Novel benzoylurea derivatives as potential antitumor agents; synthesis, activities and structure-activity relationships

  • Ki Jun Hwang*
  • , Kyung Ho Park
  • , Chong Ock Lee
  • , Beom Tae Kim
  • *Corresponding author for this work

Research output: Contribution to journalJournal articlepeer-review

Abstract

A series of pyrazoloxyphenyl benzoyl urea derivatives was designed and synthesized for cytotoxic evaluation as potential antitumor agents. The synthetic compounds were evaluated for in vitro cytotoxicity against five human tumor cell lines, including A-549, SKOV-3, SK-MEL-2, XF-498 and HCT-15. Among others, compound 11 exhibited 50∼100 times greater antitumor activities than the commercial product, Cisplatin.

Original languageEnglish
Pages (from-to)781-785
Number of pages5
JournalArchives of Pharmacal Research
Volume25
Issue number6
DOIs
StatePublished - 2002.12

UN SDGs

This output contributes to the following UN Sustainable Development Goals (SDGs)

  1. SDG 3 - Good Health and Well-being
    SDG 3 Good Health and Well-being

Keywords

  • Anticancer
  • Benzoyl Urea
  • Cisplatin
  • Cytotoxicity

Quacquarelli Symonds(QS) Subject Topics

  • Medicine
  • Engineering - Petroleum
  • Pharmacy & Pharmacology
  • Chemistry

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